Product Name: GSK-2194069

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CAT#: A-6000


  Synonym:GSK-2194069,

GSK-2194069 Chemical Structure GSK-2194069 chemical structure


IUPAC/Chemical name: 4-[4-(benzofuran-5-yl)phenyl]-3-[[(3S)-1-(cyclopropanecarbonyl)pyrrolidin-3-yl]methyl]-1H-1,2,4-triazol-5-one;2-(hydroxymethyl)-2-(methoxymethyl)quinuclidin-3-one


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Biological Activity
Potent human fatty acid synthase (hFASN) inhibitor (IC50 = 7.7 nM); inhibits hFAS β-ketoacyl reductase activity. Inhibits lipid synthesis and attenuates proliferation of A549 non-small-cell lung cancer cells (EC50 = 15 nM) in vitro.
Technical Data
M.Wt:      428.48
Formula:     C25H24N4O3
CAS#: 1332331-21-1
Purity: >99% by HPLC
Storage Conditions: 0ºC to 4 ºC for short term or -20ºC for 3 years.

Reference