Product Name: PFI-1
 CAT#: A-1288

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 Synonym:PFI-1

PFI-1 Chemical Structure
PFI-1 chemical structure


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IUPAC/Chemical name:2-​Methoxy-​N-​(3-​methyl-​2-​oxo-​1,​2,​3,​4-​tetrahydroquinazolin-​6-​yl)benzenesulfonamide

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Biological Activity
PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4. In an AlphaScreen assay it has been shown to inhibit BRD2 bromodomain 2 and BRD4 bromodomain 1 with IC₅₀ values of 98 nM and 0.22 μM, respectively.
Technical Data

Formula:C16H17N3O4S
M.Wt:347.39
CAS#:N/A
Solubility:Soluble in DMSO
Purity: >99%
Storage Conditions: 2ºC to 8 ºC, or -20ºC for 3 years.

Reference







Purchase(buy) Bromodomian and extraterninal (BET) inhibitor inhibitor PFI-1 at Active Biochem and the United State(U.S.), Germany, Japan, France,United Kingdom(UK),Switzerland, Australia distributors.