Product Name:

PHA-665752

Request
CAT#: A-1032    

Chemical Structure

Price of PHA-665752


5MG $152
10MG $300
50MG $710
We offer a substantial discount on larger orders,
please inquire via sales@activebiochem.com
or Fax: 1-201-884-1288(USA Fax#)

We match the lowest price on market.

Biological Activity

Potent, selective and ATP-competitive inhibitor of MET kinase (IC50 values are 9, 68, 200, 1400, 3000, 3800 and 6000 nM for MET, Ron, Flk-1, c-abl, FGFR1, EGFR and c-src respectively and > 10000 nM for IGF-IR, PDGFR, AURORA2, PKA, PKBα, p38α, MK2 and MK3). Antitumor agent; inhibits tumorigenicity and angiogenesis in mouse lung cancer xenografts.

Technical Data

M.Wt:      641.61
Formula:     C32H34Cl2N4O4S
Purity:     >99%
Storage Conditions :Room temperature, or -20ºC for 2 year.

Reference